Activity record

PGDB_A028267

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 60-80 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001783
PatentCN117683022A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000059
Compound IDPGDB_C000059
CompoundCC-90009;CC-90009
Source record IDPGDB_C000059
InChIKeyPWBHUSLMHZLGRN-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001783
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDCN117683022A
Compound location

CC-90009;CC-90009

CC-90009;CC-90009 enlarged structureCC-90009;CC-90009 location on patent page 5
Activity table
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