Assay

PGDB_AS001783

System: cell_basedTarget: GSPT1
Assay context summary

Assay context

21 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetGSPT1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

21 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000355
% Degradation-=60-80%1 uM-GSPT1--CN117683022APGDB_A010675PGDB_C000355PGDB_AS001783View
2D structure for PGDB_C000340
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A011973PGDB_C000340PGDB_AS001783View
2D structure for PGDB_C000348
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A013934PGDB_C000348PGDB_AS001783View
2D structure for PGDB_C000347
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A023402PGDB_C000347PGDB_AS001783View
2D structure for PGDB_C000059
% Degradation-=60-80%1 uM-GSPT1--CN117683022APGDB_A028267PGDB_C000059PGDB_AS001783View
2D structure for PGDB_C000346
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A028653PGDB_C000346PGDB_AS001783View
2D structure for PGDB_C000351
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A029276PGDB_C000351PGDB_AS001783View
2D structure for PGDB_C000350
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A030187PGDB_C000350PGDB_AS001783View
2D structure for PGDB_C000342
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A031107PGDB_C000342PGDB_AS001783View
2D structure for PGDB_C000354
% Degradation-=60-80%1 uM-GSPT1--CN117683022APGDB_A031279PGDB_C000354PGDB_AS001783View
2D structure for PGDB_C000343
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A033569PGDB_C000343PGDB_AS001783View
2D structure for PGDB_C000349
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A035893PGDB_C000349PGDB_AS001783View
2D structure for PGDB_C000356
% Degradation-=60-80%1 uM-GSPT1--CN117683022APGDB_A041441PGDB_C000356PGDB_AS001783View
2D structure for PGDB_C000358
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A042569PGDB_C000358PGDB_AS001783View
2D structure for PGDB_C000345
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A044822PGDB_C000345PGDB_AS001783View
2D structure for PGDB_C000352
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A056814PGDB_C000352PGDB_AS001783View
2D structure for PGDB_C000344
% Degradation-=30-60%1 uM-GSPT1--CN117683022APGDB_A059276PGDB_C000344PGDB_AS001783View
2D structure for PGDB_C000339
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A066242PGDB_C000339PGDB_AS001783View
2D structure for PGDB_C000357
% Degradation-=80-100%1 uM-GSPT1--CN117683022APGDB_A069738PGDB_C000357PGDB_AS001783View
2D structure for PGDB_C000341
% Degradation-=10-30%1 uM-GSPT1--CN117683022APGDB_A070340PGDB_C000341PGDB_AS001783View
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