Activity record

PGDB_A028588

Assay: % DegradationTarget: BRD4QC: standardized
Activity overview

DC50 = 10-100 nM

TargetBRD4
Assay / ReadoutWestern_blot / DC50
Assay IDPGDB_AS000558
PatentEP4605088A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C007741
Compound IDPGDB_C007741
Compound240;240
Source record IDPGDB_C007741
InChIKeyCJKQDISIQOCPNM-RTHIIRHPSA-N

Assay context

Assay IDPGDB_AS000558
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
TechnologyWestern_blot
TargetBRD4
E3Not specified

Source evidence

Patent IDEP4605088A1
Compound location

240;240

240;240 enlarged structure240;240 location on patent page 59
Activity table
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Page 195 · table middle
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