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SIMM · NJU
Assay
PGDB_AS000558
System: cell_based
Target: BRD4
Assay context summary
Assay context
30 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
BRD4
E3
Not specified
Technology
Western_blot
Activity compounds and values
Activity records
30 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
1
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A010072
PGDB_C007725
PGDB_AS000558
View
DC50
-
>
1
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A011079
PGDB_C007722
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A012397
PGDB_C007747
PGDB_AS000558
View
DC50
-
=
0.1-1
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A016101
PGDB_C007734
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A016167
PGDB_C007745
PGDB_AS000558
View
DC50
-
<
10
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A021056
PGDB_C007727
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A023510
PGDB_C007735
PGDB_AS000558
View
DC50
-
<
10
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A024033
PGDB_C007730
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A028514
PGDB_C007746
PGDB_AS000558
View
DC50
-
=
10-100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A028588
PGDB_C007741
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A030162
PGDB_C007726
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A031439
PGDB_C007750
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A031550
PGDB_C007724
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A036462
PGDB_C007739
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A036533
PGDB_C007721
PGDB_AS000558
View
DC50
-
=
0.1-1
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A039172
PGDB_C007740
PGDB_AS000558
View
DC50
-
<
100
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A040905
PGDB_C007728
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A041696
PGDB_C007749
PGDB_AS000558
View
DC50
-
<
10
nM
-
—
BRD4
-
-
EP4605088A1
PGDB_A045303
PGDB_C007731
PGDB_AS000558
View
DC50
-
>
5
uM
-
—
BRD4
-
-
EP4605088A1
PGDB_A046044
PGDB_C007752
PGDB_AS000558
View