Activity record

PGDB_A028891

Assay: % DegradationTarget: ARQC: ambiguous
Activity overview

degradation = 50 %

TargetAR
Cell lineLNCaP
Concentration5 uM
Assay / Readout% Degradation
Assay IDPGDB_AS002019
PatentJP5998117B2
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C026012
Compound IDPGDB_C026012
CompoundASC-Q111
Source record IDPGDB_C026012
InChIKeyXQLWYXLCJXPOMJ-ANOAMAFRSA-N

Assay context

Assay IDPGDB_AS002019
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration5 uM
Detection targetprotein_degradation
TargetAR
E3Not specified
Cell lineLNCaP
OrganismHomo sapiens

Source evidence

Patent IDJP5998117B2
Compound location

ASC-Q111

ASC-Q111 enlarged structureASC-Q111 location on patent page 61
Activity table
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