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SIMM · NJU
Assay
PGDB_AS002019
System: cell_based
Cell line: LNCaP
Assay context summary
Assay context
11 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
E3
Not specified
Cell line
LNCaP
Organism
Homo sapiens
Detection target
protein_degradation
Activity compounds and values
Activity records
11 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
27
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A008995
PGDB_C026008
PGDB_AS002019
View
% Degradation
-
=
58
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A027804
PGDB_C026011
PGDB_AS002019
View
% Degradation
-
=
50
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A028891
PGDB_C026012
PGDB_AS002019
View
% Degradation
-
=
43
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A033766
PGDB_C026016
PGDB_AS002019
View
% Degradation
-
=
73
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A037265
PGDB_C026007
PGDB_AS002019
View
% Degradation
-
=
6
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A042292
PGDB_C026009
PGDB_AS002019
View
% Degradation
-
=
47
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A056270
PGDB_C026005
PGDB_AS002019
View
% Degradation
-
=
30
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A057250
PGDB_C026014
PGDB_AS002019
View
% Degradation
-
=
14
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A071762
PGDB_C026010
PGDB_AS002019
View
% Degradation
-
=
81
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A075110
PGDB_C026015
PGDB_AS002019
View
% Degradation
-
=
74
%
5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A077154
PGDB_C026017
PGDB_AS002019
View