Activity record

PGDB_A030086

Assay: biochemicalQC: ambiguous
Activity overview

selectivity_index = 3.2 fold

Time60 min
ControlCDK7 / CDK12
Assay / ReadoutFold change / biochemical
Assay IDPGDB_AS002236
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006580
Compound IDPGDB_C006580
CompoundH-APPAMP-013;H-APPAMP-013
Source record IDPGDB_C006580
InChIKeyBZQQJGZLMVFPHN-GCJKJVERSA-N

Assay context

Assay IDPGDB_AS002236
Assay familybiochemical
Assay systembiochemical
ReadoutFold change
Treatment time60 min
TargetCDK12 | CDK7
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-013;H-APPAMP-013

H-APPAMP-013;H-APPAMP-013 enlarged structureH-APPAMP-013;H-APPAMP-013 location on patent page 39
Activity table
Page 195 · table start
Page 196 · table middle
Page 197 · table end