Activity record

PGDB_A030140

Assay: bindingTarget: CRBNQC: standardized
Activity overview

IC50 > 1700 nM

TargetCRBN
E3 ligaseCRBN
Time12 h
Assay / Readoutfluorescence / IC50
Assay IDPGDB_AS000438
PatentWO2022219412A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C026003
Compound IDPGDB_C026003
Compound18
Source record IDPGDB_C001734
InChIKeyBOYRHANJCVXPEM-VWLOTQADSA-N

Assay context

Assay IDPGDB_AS000438
Assay familybinding
Assay systembiochemical
ReadoutIC50
Technologyfluorescence
Treatment time12 h
TargetCRBN
E3CRBN

Source evidence

Patent IDWO2022219412A1
Activity table
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