Activity record

PGDB_A031087

Assay: bindingTarget: CRBNQC: standardized
Activity overview

Ki = 1-5 uM

TargetCRBN
E3 ligaseCRBN
Time60 min
Assay / Readoutfluorescence / Ki
Assay IDPGDB_AS002364
PatentWO2022146151A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009609
Compound IDPGDB_C009609
Compound{277}
Source record IDPGDB_C009609
InChIKeyPOYGFAYCNOFXKY-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002364
Assay familybinding
Assay systembiochemical
ReadoutKi
Technologyfluorescence
Treatment time60 min
TargetCRBN | DDB1
E3CRBN | DDB1

Source evidence

Patent IDWO2022146151A1
Activity table
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