Assay

PGDB_AS002364

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

25 activity records
Assay familybinding
Systembiochemical
ReadoutKi
TargetCRBN | DDB1
E3CRBN | DDB1
Technologyfluorescence
Activity compounds and values

Activity records

25 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C009603
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A008671PGDB_C009603PGDB_AS002364View
2D structure for PGDB_C008731
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A011992PGDB_C008731PGDB_AS002364View
2D structure for PGDB_C009611
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A012536PGDB_C009611PGDB_AS002364View
2D structure for PGDB_C009610
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A013255PGDB_C009610PGDB_AS002364View
2D structure for PGDB_C009616
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A014071PGDB_C009616PGDB_AS002364View
2D structure for PGDB_C009617
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A015276PGDB_C009617PGDB_AS002364View
2D structure for PGDB_C009619
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A020502PGDB_C009619PGDB_AS002364View
2D structure for PGDB_C009622
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A022447PGDB_C009622PGDB_AS002364View
2D structure for PGDB_C019024
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A026969PGDB_C019024PGDB_AS002364View
2D structure for PGDB_C009608
Ki-=5-10uM-—CRBNCRBN-WO2022146151A1PGDB_A030799PGDB_C009608PGDB_AS002364View
2D structure for PGDB_C009609
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A031087PGDB_C009609PGDB_AS002364View
2D structure for PGDB_C009614
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A033268PGDB_C009614PGDB_AS002364View
2D structure for PGDB_C009613
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A034019PGDB_C009613PGDB_AS002364View
2D structure for PGDB_C009601
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A034274PGDB_C009601PGDB_AS002364View
2D structure for PGDB_C009623
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A037695PGDB_C009623PGDB_AS002364View
2D structure for PGDB_C009604
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A039091PGDB_C009604PGDB_AS002364View
2D structure for PGDB_C009602
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A042777PGDB_C009602PGDB_AS002364View
2D structure for PGDB_C009612
Ki-<=1uM-—CRBNCRBN-WO2022146151A1PGDB_A049598PGDB_C009612PGDB_AS002364View
2D structure for PGDB_C009615
Ki-=1-5uM-—CRBNCRBN-WO2022146151A1PGDB_A053100PGDB_C009615PGDB_AS002364View
2D structure for PGDB_C009607
Ki-=5-10uM-—CRBNCRBN-WO2022146151A1PGDB_A059547PGDB_C009607PGDB_AS002364View
Page 1 of 2 · 25 records