Activity record

PGDB_A034267

Assay: % DegradationTarget: CSNK1A1QC: ambiguous
Activity overview

degradation = 63.3 %

TargetCSNK1A1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS000685
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002818
Compound IDPGDB_C002818
Compound59;59;59
Source record IDPGDB_C002818
InChIKeyGRDLGPVCCSHERU-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000685
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetCSNK1A1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

59;59;59

59;59;59 enlarged structure59;59;59 location on patent page 9
Activity table
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