Assay

PGDB_AS000685

System: cell_basedTarget: CSNK1A1
Assay context summary

Assay context

44 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetCSNK1A1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

44 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002810
% Degradation-=67.4%1 uM-CSNK1A1--WO2024059107A1PGDB_A007173PGDB_C002810PGDB_AS000685View
2D structure for PGDB_C002813
% Degradation-=55.4%1 uM-CSNK1A1--WO2024059107A1PGDB_A008181PGDB_C002813PGDB_AS000685View
2D structure for PGDB_C002829
% Degradation-=69.9%1 uM-CSNK1A1--WO2024059107A1PGDB_A009809PGDB_C002829PGDB_AS000685View
2D structure for PGDB_C002842
% Degradation-=80.3%1 uM-CSNK1A1--WO2024059107A1PGDB_A010735PGDB_C002842PGDB_AS000685View
2D structure for PGDB_C002821
% Degradation-=57%1 uM-CSNK1A1--WO2024059107A1PGDB_A010956PGDB_C002821PGDB_AS000685View
2D structure for PGDB_C002845
% Degradation-=71.5%1 uM-CSNK1A1--WO2024059107A1PGDB_A013121PGDB_C002845PGDB_AS000685View
2D structure for PGDB_C002838
% Degradation-=72%1 uM-CSNK1A1--WO2024059107A1PGDB_A014173PGDB_C002838PGDB_AS000685View
2D structure for PGDB_C002806
% Degradation-=65.5%1 uM-CSNK1A1--WO2024059107A1PGDB_A019793PGDB_C002806PGDB_AS000685View
2D structure for PGDB_C002830
% Degradation-=60.4%1 uM-CSNK1A1--WO2024059107A1PGDB_A022650PGDB_C002830PGDB_AS000685View
2D structure for PGDB_C002835
% Degradation-=64.8%1 uM-CSNK1A1--WO2024059107A1PGDB_A024568PGDB_C002835PGDB_AS000685View
2D structure for PGDB_C002809
% Degradation-=67%1 uM-CSNK1A1--WO2024059107A1PGDB_A025242PGDB_C002809PGDB_AS000685View
2D structure for PGDB_C002833
% Degradation-=38.1%1 uM-CSNK1A1--WO2024059107A1PGDB_A026122PGDB_C002833PGDB_AS000685View
2D structure for PGDB_C002843
% Degradation-=80.1%1 uM-CSNK1A1--WO2024059107A1PGDB_A027404PGDB_C002843PGDB_AS000685View
2D structure for PGDB_C002831
% Degradation-=66.9%1 uM-CSNK1A1--WO2024059107A1PGDB_A028709PGDB_C002831PGDB_AS000685View
2D structure for PGDB_C002834
% Degradation-=69.5%1 uM-CSNK1A1--WO2024059107A1PGDB_A030934PGDB_C002834PGDB_AS000685View
2D structure for PGDB_C002815
% Degradation-=56.9%1 uM-CSNK1A1--WO2024059107A1PGDB_A031166PGDB_C002815PGDB_AS000685View
2D structure for PGDB_C002812
% Degradation-=69.8%1 uM-CSNK1A1--WO2024059107A1PGDB_A031991PGDB_C002812PGDB_AS000685View
2D structure for PGDB_C002818
% Degradation-=63.3%1 uM-CSNK1A1--WO2024059107A1PGDB_A034267PGDB_C002818PGDB_AS000685View
2D structure for PGDB_C002817
% Degradation-=60.3%1 uM-CSNK1A1--WO2024059107A1PGDB_A034940PGDB_C002817PGDB_AS000685View
2D structure for PGDB_C002849
% Degradation-=41.2%1 uM-CSNK1A1--WO2024059107A1PGDB_A035299PGDB_C002849PGDB_AS000685View
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