Activity record

PGDB_A035892

Assay: % DegradationQC: standardized
Activity overview

degradation = 70-90 %

Cell lineMOLM-13
Assay / Readout% Degradation
Assay IDPGDB_AS002573
PatentCN117756818A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000379
Compound IDPGDB_C000379
CompounddBET6
Source record IDPGDB_C000379
InChIKeyJGQPZPLJOBHHBK-UFXYQILXSA-N

Assay context

Assay IDPGDB_AS002573
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Detection targetprotein_degradation
TargetBRD4
E3Not specified
Cell lineMOLM-13
OrganismHomo sapiens

Source evidence

Patent IDCN117756818A
Compound location

dBET6

dBET6 enlarged structuredBET6 location on patent page 18
Activity table
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