Activity record

PGDB_A036533

Assay: % DegradationTarget: BRD4QC: standardized
Activity overview

DC50 < 100 nM

TargetBRD4
Assay / ReadoutWestern_blot / DC50
Assay IDPGDB_AS000558
PatentEP4605088A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C007721
Compound IDPGDB_C007721
Compound140;140;140
Source record IDPGDB_C007721
InChIKeyMEWPHCREUNWPJB-ODUIWNOOSA-N

Assay context

Assay IDPGDB_AS000558
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
TechnologyWestern_blot
TargetBRD4
E3Not specified

Source evidence

Patent IDEP4605088A1
Compound location

140;140;140

140;140;140 enlarged structure140;140;140 location on patent page 49
Activity table
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Page 195 · table middle
Page 196 · table end