Activity record

PGDB_A042569

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 30-60 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001783
PatentCN117683022A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000358
Compound IDPGDB_C000358
Compound20;20
Source record IDPGDB_C000358
InChIKeyTZRQQGHBPSJZSZ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001783
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDCN117683022A
Compound location

20;20

20;20 enlarged structure20;20 location on patent page 3
Activity table
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