Activity record

PGDB_A044821

Assay: biochemicalTarget: CDK12QC: ambiguous
Activity overview

IC50 = 50.2 nM

TargetCDK12
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS001187
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006570
Compound IDPGDB_C006570
CompoundH-APPAMP-003;H-APPAMP-003
Source record IDPGDB_C006570
InChIKeyJWLYZTFPPDFIIV-APWZRJJASA-N

Assay context

Assay IDPGDB_AS001187
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK12
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-003;H-APPAMP-003

H-APPAMP-003;H-APPAMP-003 enlarged structureH-APPAMP-003;H-APPAMP-003 location on patent page 37
Activity table
Page 195 · table start
Page 196 · table middle
Page 197 · table end