Assay

PGDB_AS001187

System: biochemicalTarget: CDK12
Assay context summary

Assay context

48 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCDK12
E3Not specified
OrganismHomo sapiens
Activity compounds and values

Activity records

48 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006566
IC50-=253nM-—CDK12--CN114929708BPGDB_A008142PGDB_C006566PGDB_AS001187View
2D structure for PGDB_C006608
IC50-=46nM-—CDK12--CN114929708BPGDB_A010565PGDB_C006608PGDB_AS001187View
2D structure for PGDB_C006567
IC50-=597nM-—CDK12--CN114929708BPGDB_A011106PGDB_C006567PGDB_AS001187View
2D structure for PGDB_C006596
IC50-=65nM-—CDK12--CN114929708BPGDB_A011587PGDB_C006596PGDB_AS001187View
2D structure for PGDB_C006607
IC50-=48nM-—CDK12--CN114929708BPGDB_A012216PGDB_C006607PGDB_AS001187View
2D structure for PGDB_C006595
IC50-=37nM-—CDK12--CN114929708BPGDB_A014674PGDB_C006595PGDB_AS001187View
2D structure for PGDB_C006579
IC50-=26nM-—CDK12--CN114929708BPGDB_A015263PGDB_C006579PGDB_AS001187View
2D structure for PGDB_C006565
IC50-=3200nM-—CDK12--CN114929708BPGDB_A016022PGDB_C006565PGDB_AS001187View
2D structure for PGDB_C006598
IC50-=24nM-—CDK12--CN114929708BPGDB_A017367PGDB_C006598PGDB_AS001187View
2D structure for PGDB_C006599
IC50-=45nM-—CDK12--CN114929708BPGDB_A022602PGDB_C006599PGDB_AS001187View
2D structure for PGDB_C006578
IC50-=33nM-—CDK12--CN114929708BPGDB_A022914PGDB_C006578PGDB_AS001187View
2D structure for PGDB_C006604
IC50-=208nM-—CDK12--CN114929708BPGDB_A023580PGDB_C006604PGDB_AS001187View
2D structure for PGDB_C006584
IC50-=63nM-—CDK12--CN114929708BPGDB_A024674PGDB_C006584PGDB_AS001187View
2D structure for PGDB_C006568
IC50-=38nM-—CDK12--CN114929708BPGDB_A025942PGDB_C006568PGDB_AS001187View
2D structure for PGDB_C006569
IC50-=71.5nM-—CDK12--CN114929708BPGDB_A026690PGDB_C006569PGDB_AS001187View
2D structure for PGDB_C006580
IC50-=70nM-—CDK12--CN114929708BPGDB_A027116PGDB_C006580PGDB_AS001187View
2D structure for PGDB_C006577
IC50-=40nM-—CDK12--CN114929708BPGDB_A027173PGDB_C006577PGDB_AS001187View
2D structure for PGDB_C006573
IC50-=26.9nM-—CDK12--CN114929708BPGDB_A027345PGDB_C006573PGDB_AS001187View
2D structure for PGDB_C006585
IC50-=65nM-—CDK12--CN114929708BPGDB_A027574PGDB_C006585PGDB_AS001187View
2D structure for PGDB_C006611
IC50-=40nM-—CDK12--CN114929708BPGDB_A029553PGDB_C006611PGDB_AS001187View
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