PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Loading activity
Loading detail record from the SQLite release...
PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Activity record
PGDB_A046816
Assay: % Degradation
Target: CRBN
QC: standardized
Activity overview
degradation = 31.99 %
Target
CRBN
E3 ligase
CRBN
Concentration
Concentration series: 10 nM, 10 uM
Assay / Readout
Western_blot / % Degradation
Assay ID
PGDB_AS002247
Patent
US20220362229A1
QC status
standardized
Evidence details
Compound, assay context, and source
Compound
Compound ID
PGDB_C009092
Compound
{606} EC1-151 M.W. = 670.72
Source record ID
PGDB_C009092
InChIKey
OOVOAMUEWLDPIX-UHFFFAOYSA-N
Assay context
Assay ID
PGDB_AS002247
Assay family
% Degradation
Assay system
cell_based
Readout
% Degradation
Technology
Western_blot
Concentration
Concentration series: 10 nM, 10 uM
Detection target
protein_degradation
Target
CRBN
E3
CRBN
Source evidence
Patent ID
US20220362229A1
Activity table