Activity record

PGDB_A049718

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

inhibition = 91.87 %

TargetGSPT1
Cell lineNCI-H1581
Time3 d
Assay / Readoutluminescence / % Inhibition
Assay IDPGDB_AS000288
PatentWO2023001028A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C001867
Compound IDPGDB_C001867
CompoundWX015
Source record IDPGDB_C001867
InChIKeyUSEQRCHYCVHABT-SFHVURJKSA-N

Assay context

Assay IDPGDB_AS000288
Assay familyviability
Assay systemcell_based
Readout% Inhibition
Technologyluminescence
Treatment time3 d
Detection targetcell_inhibition
TargetGSPT1
E3Not specified
Cell lineNCI-H1581

Source evidence

Patent IDWO2023001028A1
Compound location

WX015

WX015 enlarged structureWX015 location on patent page 39
Activity table
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