Activity record

PGDB_A052245

Assay: cellular_functionTarget: ESR1QC: ambiguous
Activity overview

IC50 = 4.9 nM

TargetESR1
Cell lineHEK293
Time20 h
Assay / Readoutfluorescence / IC50
Assay IDPGDB_AS000727
PatentCN115260206A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006618
Compound IDPGDB_C006618
Compound化合物8;实施例8;实施例8
Source record IDPGDB_C006618
InChIKeyUPDGUCDCSDPSRG-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000727
Assay familycellular_function
Assay systemcell_based
ReadoutIC50
Technologyfluorescence
Treatment time20 h
TargetESR1
E3Not specified
Cell lineHEK293

Source evidence

Patent IDCN115260206A
Compound location

化合物8;实施例8;实施例8

化合物8;实施例8;实施例8 enlarged structure化合物8;实施例8;实施例8 location on patent page 19
Activity table
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