Activity record

PGDB_A052247

Assay: bindingQC: standardized_posthoc
Activity overview

selectivity_index = 100-500 fold

ControlCDK2 / CDK12
Assay / ReadoutFold change / binding
Assay IDPGDB_AS002325
PatentWO2025110815A1
QC statusstandardized_posthoc
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010984
Compound IDPGDB_C010984
Compound46
Source record IDPGDB_C010984
InChIKeyUGGUYTVWTNWSPB-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002325
Assay familybinding
Assay systemcell_based
ReadoutFold change
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

46

46 enlarged structure46 location on patent page 98
Activity table
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