PatGlueDB | Molecular Glue Patent Bioactivity Database

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35 activity records

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Systemcell_based

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E3Not specified

Activity compounds and values

Activity records

35 records

Metric	Control	Relation	Value	Unit	Concentration	Time	Target	E3	Cell line	Patent	Record ID	Compound	Assay	Details
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A011011	PGDB_C010959	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	<=	100	fold	-	—	-	-	-	WO2025110815A1	PGDB_A011851	PGDB_C010951	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	<=	100	fold	-	—	-	-	-	WO2025110815A1	PGDB_A016052	PGDB_C010917	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A016073	PGDB_C010944	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A017436	PGDB_C010960	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A021921	PGDB_C010956	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A023313	PGDB_C010944	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	<=	100	fold	-	—	-	-	-	WO2025110815A1	PGDB_A025176	PGDB_C010919	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A026320	PGDB_C010952	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A028852	PGDB_C010956	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A030421	PGDB_C010984	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A031377	PGDB_C010955	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A033382	PGDB_C011002	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A038429	PGDB_C010960	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A043004	PGDB_C010920	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A043160	PGDB_C010955	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	<=	100	fold	-	—	-	-	-	WO2025110815A1	PGDB_A045492	PGDB_C010951	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A046428	PGDB_C010916	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	=	100-500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A046907	PGDB_C010914	PGDB_AS002325	View
Selectivity index	CDK2 / CDK12	>	500	fold	-	—	-	-	-	WO2025110815A1	PGDB_A047044	PGDB_C010958	PGDB_AS002325	View

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