Activity record

PGDB_A053491

Assay: viabilityTarget: CDK12QC: ambiguous
Activity overview

IC50 = 7.3 nM

TargetCDK12
Cell lineA673
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS002570
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006581
Compound IDPGDB_C006581
CompoundH-APPAMP-014;H-APPAMP-014
Source record IDPGDB_C006581
InChIKeyGURJFCBCOPFZHK-GCJKJVERSA-N

Assay context

Assay IDPGDB_AS002570
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified
Cell lineA673

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-014;H-APPAMP-014

H-APPAMP-014;H-APPAMP-014 enlarged structureH-APPAMP-014;H-APPAMP-014 location on patent page 39
Activity table
Page 198 · table start
Page 199 · table end