Activity record

PGDB_A054627

Assay: bindingQC: standardized_posthoc
Activity overview

selectivity_index > 500 fold

ControlCDK2 / CDK12
Assay / ReadoutFold change / binding
Assay IDPGDB_AS002325
PatentWO2025110815A1
QC statusstandardized_posthoc
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010921
Compound IDPGDB_C010921
Compound18
Source record IDPGDB_C010921
InChIKeyBGSTVVYHLREGKP-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002325
Assay familybinding
Assay systemcell_based
ReadoutFold change
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

18

18 enlarged structure18 location on patent page 75
Activity table
Page 154 · table start