Activity record

PGDB_A056503

Assay: biochemicalQC: manual_curated
Activity overview

selectivity_index = 100-500 fold

Time120 min
ControlCDK1 / CDK12
Assay / Readoutselectivity_fold / biochemical
Assay IDPGDB_AS002417
PatentWO2025110815A1
QC statusmanual_curated
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010954
Compound IDPGDB_C010954
Compound71
Source record IDPGDB_C010954
InChIKeyMQSLRPFFONOQCJ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002417
Assay familybiochemical
Assay systembiochemical
Readoutselectivity_fold
Treatment time120 min
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

71

71 enlarged structure71 location on patent page 115
Activity table
Page 154 · table start