Activity record

PGDB_A058325

Assay: % DegradationTarget: CDK12QC: ambiguous
Activity overview

IC50 <= 0.1 uM

TargetCDK12
Assay / ReadoutIC50 / % Degradation
Assay IDPGDB_AS002095
PatentWO2025110815A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010916
Compound IDPGDB_C010916
Compound13
Source record IDPGDB_C010916
InChIKeyFDLFTAYEXIHQOV-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002095
Assay family% Degradation
Assay systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

13

13 enlarged structure13 location on patent page 74
Activity table
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