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SIMM · NJU
Assay
PGDB_AS002095
System: cell_based
Assay context summary
Assay context
108 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
E3
Not specified
Activity compounds and values
Activity records
108 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A007735
PGDB_C010941
PGDB_AS002095
View
IC50
-
>
0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A010380
PGDB_C010927
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A010555
PGDB_C010962
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A011164
PGDB_C010912
PGDB_AS002095
View
IC50
-
>
0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A011385
PGDB_C010973
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A012233
PGDB_C010965
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A014548
PGDB_C010971
PGDB_AS002095
View
IC50
-
=
0.1-0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A014823
PGDB_C010909
PGDB_AS002095
View
IC50
-
=
0.1-0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A015141
PGDB_C010908
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A016888
PGDB_C010953
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A018860
PGDB_C010940
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A019068
PGDB_C010905
PGDB_AS002095
View
IC50
-
>
0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A019091
PGDB_C010975
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A019915
PGDB_C010920
PGDB_AS002095
View
IC50
-
>
0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A020174
PGDB_C010937
PGDB_AS002095
View
IC50
-
=
0.1-0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A020842
PGDB_C010985
PGDB_AS002095
View
IC50
-
=
0.1-0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A021100
PGDB_C010917
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A021678
PGDB_C010997
PGDB_AS002095
View
IC50
-
<=
0.1
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A022133
PGDB_C010994
PGDB_AS002095
View
IC50
-
=
0.1-0.5
uM
-
—
CDK12
-
-
WO2025110815A1
PGDB_A022310
PGDB_C010896
PGDB_AS002095
View