Assay context summary

Assay context

108 activity records
Activity compounds and values

Activity records

108 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C010941
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A007735PGDB_C010941PGDB_AS002095View
2D structure for PGDB_C010927
IC50->0.5uM-CDK12--WO2025110815A1PGDB_A010380PGDB_C010927PGDB_AS002095View
2D structure for PGDB_C010962
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A010555PGDB_C010962PGDB_AS002095View
2D structure for PGDB_C010912
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A011164PGDB_C010912PGDB_AS002095View
2D structure for PGDB_C010973
IC50->0.5uM-CDK12--WO2025110815A1PGDB_A011385PGDB_C010973PGDB_AS002095View
2D structure for PGDB_C010965
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A012233PGDB_C010965PGDB_AS002095View
2D structure for PGDB_C010971
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A014548PGDB_C010971PGDB_AS002095View
2D structure for PGDB_C010909
IC50-=0.1-0.5uM-CDK12--WO2025110815A1PGDB_A014823PGDB_C010909PGDB_AS002095View
2D structure for PGDB_C010908
IC50-=0.1-0.5uM-CDK12--WO2025110815A1PGDB_A015141PGDB_C010908PGDB_AS002095View
2D structure for PGDB_C010953
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A016888PGDB_C010953PGDB_AS002095View
2D structure for PGDB_C010940
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A018860PGDB_C010940PGDB_AS002095View
2D structure for PGDB_C010905
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A019068PGDB_C010905PGDB_AS002095View
2D structure for PGDB_C010975
IC50->0.5uM-CDK12--WO2025110815A1PGDB_A019091PGDB_C010975PGDB_AS002095View
2D structure for PGDB_C010920
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A019915PGDB_C010920PGDB_AS002095View
2D structure for PGDB_C010937
IC50->0.5uM-CDK12--WO2025110815A1PGDB_A020174PGDB_C010937PGDB_AS002095View
2D structure for PGDB_C010985
IC50-=0.1-0.5uM-CDK12--WO2025110815A1PGDB_A020842PGDB_C010985PGDB_AS002095View
2D structure for PGDB_C010917
IC50-=0.1-0.5uM-CDK12--WO2025110815A1PGDB_A021100PGDB_C010917PGDB_AS002095View
2D structure for PGDB_C010997
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A021678PGDB_C010997PGDB_AS002095View
2D structure for PGDB_C010994
IC50-<=0.1uM-CDK12--WO2025110815A1PGDB_A022133PGDB_C010994PGDB_AS002095View
2D structure for PGDB_C010896
IC50-=0.1-0.5uM-CDK12--WO2025110815A1PGDB_A022310PGDB_C010896PGDB_AS002095View