Activity record

PGDB_A059988

Assay: biochemicalTarget: CDK12QC: ambiguous
Activity overview

IC50 = 208 nM

TargetCDK12
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS001268
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006604
Compound IDPGDB_C006604
CompoundH-APPAMP-037
Source record IDPGDB_C006604
InChIKeyCDYKZMBMURUOQF-QAPCUYQASA-N

Assay context

Assay IDPGDB_AS001268
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK12
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-037

H-APPAMP-037 enlarged structureH-APPAMP-037 location on patent page 45
Activity table
Page 198 · table start
Page 199 · table end