Assay

PGDB_AS001268

System: biochemicalTarget: CDK12
Assay context summary

Assay context

45 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCDK12
E3Not specified
OrganismHomo sapiens
Activity compounds and values

Activity records

45 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006612
IC50-=18nM-—CDK12--CN114929708BPGDB_A007206PGDB_C006612PGDB_AS001268View
2D structure for PGDB_C006595
IC50-=37nM-—CDK12--CN114929708BPGDB_A007534PGDB_C006595PGDB_AS001268View
2D structure for PGDB_C006609
IC50-=100nM-—CDK12--CN114929708BPGDB_A008731PGDB_C006609PGDB_AS001268View
2D structure for PGDB_C006608
IC50-=46nM-—CDK12--CN114929708BPGDB_A010708PGDB_C006608PGDB_AS001268View
2D structure for PGDB_C006576
IC50-=38nM-—CDK12--CN114929708BPGDB_A011096PGDB_C006576PGDB_AS001268View
2D structure for PGDB_C006570
IC50-=50nM-—CDK12--CN114929708BPGDB_A012281PGDB_C006570PGDB_AS001268View
2D structure for PGDB_C006606
IC50-=48nM-—CDK12--CN114929708BPGDB_A013039PGDB_C006606PGDB_AS001268View
2D structure for PGDB_C006594
IC50-=28nM-—CDK12--CN114929708BPGDB_A013193PGDB_C006594PGDB_AS001268View
2D structure for PGDB_C006585
IC50-=65nM-—CDK12--CN114929708BPGDB_A014165PGDB_C006585PGDB_AS001268View
2D structure for PGDB_C006582
IC50-=277nM-—CDK12--CN114929708BPGDB_A014945PGDB_C006582PGDB_AS001268View
2D structure for PGDB_C006590
IC50-=702nM-—CDK12--CN114929708BPGDB_A015003PGDB_C006590PGDB_AS001268View
2D structure for PGDB_C006607
IC50-=48nM-—CDK12--CN114929708BPGDB_A020921PGDB_C006607PGDB_AS001268View
2D structure for PGDB_C006589
IC50-=164nM-—CDK12--CN114929708BPGDB_A022014PGDB_C006589PGDB_AS001268View
2D structure for PGDB_C006593
IC50-=31nM-—CDK12--CN114929708BPGDB_A022399PGDB_C006593PGDB_AS001268View
2D structure for PGDB_C006601
IC50-=173nM-—CDK12--CN114929708BPGDB_A030210PGDB_C006601PGDB_AS001268View
2D structure for PGDB_C006597
IC50-=75nM-—CDK12--CN114929708BPGDB_A030407PGDB_C006597PGDB_AS001268View
2D structure for PGDB_C006611
IC50-=40nM-—CDK12--CN114929708BPGDB_A034513PGDB_C006611PGDB_AS001268View
2D structure for PGDB_C006584
IC50-=143nM-—CDK12--CN114929708BPGDB_A037493PGDB_C006584PGDB_AS001268View
2D structure for PGDB_C006580
IC50-=70nM-—CDK12--CN114929708BPGDB_A037825PGDB_C006580PGDB_AS001268View
2D structure for PGDB_C006569
IC50-=71nM-—CDK12--CN114929708BPGDB_A037974PGDB_C006569PGDB_AS001268View
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