Activity record

PGDB_A060235

Assay: biochemicalTarget: CDK12QC: ambiguous
Activity overview

IC50 = 18 nM

TargetCDK12
Time60 min
Assay / ReadoutIC50 / biochemical
Assay IDPGDB_AS001066
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006612
Compound IDPGDB_C006612
CompoundH-APPAMP-045;H-APPAMP-045
Source record IDPGDB_C006612
InChIKeyRPJBXXVLFGLSLU-RDGATRHJSA-N

Assay context

Assay IDPGDB_AS001066
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
Treatment time60 min
TargetCDK12
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-045;H-APPAMP-045

H-APPAMP-045;H-APPAMP-045 enlarged structureH-APPAMP-045;H-APPAMP-045 location on patent page 47
Activity table
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