Assay
PGDB_AS001066
System: biochemicalTarget: CDK12
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | IC50 | - | = | 55 | nM | - | — | CDK12 | - | - | CN114929708B | PGDB_A010600 | PGDB_C006571 | PGDB_AS001066 | View |
 | IC50 | - | = | 36 | nM | - | — | CDK12 | - | - | CN114929708B | PGDB_A028881 | PGDB_C006592 | PGDB_AS001066 | View |
 | IC50 | - | = | 40 | nM | - | — | CDK12 | - | - | CN114929708B | PGDB_A039571 | PGDB_C006611 | PGDB_AS001066 | View |
 | IC50 | - | = | 21 | nM | - | — | CDK12 | - | - | CN114929708B | PGDB_A051861 | PGDB_C006610 | PGDB_AS001066 | View |
 | IC50 | - | = | 18 | nM | - | — | CDK12 | - | - | CN114929708B | PGDB_A060235 | PGDB_C006612 | PGDB_AS001066 | View |