Activity record

PGDB_A061449

Assay: % DegradationTarget: MYCQC: ambiguous
Activity overview

degradation = 82.14 %

TargetMYC
Cell lineDaudi
Concentration7.5 uM
Time12 h
Assay / Readout% Degradation
Assay IDPGDB_AS000998
PatentCN120040371B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C007049
Compound IDPGDB_C007049
Compound实施例28
Source record IDPGDB_C007049
InChIKeyKGRIPICRCPSHLC-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000998
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration7.5 uM
Treatment time12 h
Detection targetprotein_degradation
TargetMYC
E3Not specified
Cell lineDaudi

Source evidence

Patent IDCN120040371B
Compound location

实施例28

实施例28 enlarged structure实施例28 location on patent page 18
Activity table
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