Activity record

PGDB_A062230

Assay: viabilityTarget: BTKQC: standardized
Activity overview

IC50 = 500-1000 nM

TargetBTK
Cell lineVCaP
Time96 h
Assay / ReadoutCCK-8 / viability
Assay IDPGDB_AS001439
PatentCN116239566A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C025804
Compound IDPGDB_C025804
CompoundGT-03552
Source record IDPGDB_C015974
InChIKeyJWYUUNPRUQXJEQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001439
Assay familyviability
Assay systemcell_based
Readoutviability
TechnologyCCK-8
Treatment time96 h
Detection target% Cell viability
TargetBTK
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDCN116239566A
Compound location

GT-03552

GT-03552 enlarged structureGT-03552 location on patent page 266
Activity table
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