Assay
PGDB_AS001439
System: cell_basedCell line: VCaP
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A009236 | PGDB_C025807 | PGDB_AS001439 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A016789 | PGDB_C025803 | PGDB_AS001439 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A019853 | PGDB_C015982 | PGDB_AS001439 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A021909 | PGDB_C025806 | PGDB_AS001439 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A042119 | PGDB_C025814 | PGDB_AS001439 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A052616 | PGDB_C025808 | PGDB_AS001439 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | BTK | - | VCaP | CN116239566A | PGDB_A062230 | PGDB_C025804 | PGDB_AS001439 | View |