Activity record

PGDB_A066961

Assay: % DegradationTarget: CSNK1A1QC: ambiguous
Activity overview

degradation = 76.5 %

TargetCSNK1A1
Concentration100 nM
Assay / Readout% Degradation
Assay IDPGDB_AS000209
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002846
Compound IDPGDB_C002846
Compound95;95;95
Source record IDPGDB_C002846
InChIKeyNBFAWLWAYOGJOI-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000209
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration100 nM
Detection targetprotein_degradation
TargetCSNK1A1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

95;95;95

95;95;95 enlarged structure95;95;95 location on patent page 12
Activity table
Page 141 · table single