Assay

PGDB_AS000209

System: cell_basedTarget: CSNK1A1
Assay context summary

Assay context

44 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetCSNK1A1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

44 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002819
% Degradation-=50.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A009085PGDB_C002819PGDB_AS000209View
2D structure for PGDB_C002843
% Degradation-=76.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A009175PGDB_C002843PGDB_AS000209View
2D structure for PGDB_C002828
% Degradation-=48.1%100 nM-CSNK1A1--WO2024059107A1PGDB_A009504PGDB_C002828PGDB_AS000209View
2D structure for PGDB_C002845
% Degradation-=51.3%100 nM-CSNK1A1--WO2024059107A1PGDB_A010007PGDB_C002845PGDB_AS000209View
2D structure for PGDB_C002813
% Degradation-=36.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A011755PGDB_C002813PGDB_AS000209View
2D structure for PGDB_C002849
% Degradation-=18.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A012154PGDB_C002849PGDB_AS000209View
2D structure for PGDB_C002814
% Degradation-=33.5%100 nM-CSNK1A1--WO2024059107A1PGDB_A012158PGDB_C002814PGDB_AS000209View
2D structure for PGDB_C002809
% Degradation-=60.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A020835PGDB_C002809PGDB_AS000209View
2D structure for PGDB_C002820
% Degradation-=33.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A021463PGDB_C002820PGDB_AS000209View
2D structure for PGDB_C002840
% Degradation-=46.5%100 nM-CSNK1A1--WO2024059107A1PGDB_A023142PGDB_C002840PGDB_AS000209View
2D structure for PGDB_C002815
% Degradation-=51.1%100 nM-CSNK1A1--WO2024059107A1PGDB_A024114PGDB_C002815PGDB_AS000209View
2D structure for PGDB_C002835
% Degradation-=59.5%100 nM-CSNK1A1--WO2024059107A1PGDB_A025646PGDB_C002835PGDB_AS000209View
2D structure for PGDB_C002847
% Degradation-=9.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A027621PGDB_C002847PGDB_AS000209View
2D structure for PGDB_C002825
% Degradation-=40.3%100 nM-CSNK1A1--WO2024059107A1PGDB_A029419PGDB_C002825PGDB_AS000209View
2D structure for PGDB_C002831
% Degradation-=63.5%100 nM-CSNK1A1--WO2024059107A1PGDB_A031383PGDB_C002831PGDB_AS000209View
2D structure for PGDB_C002833
% Degradation-=59.4%100 nM-CSNK1A1--WO2024059107A1PGDB_A031478PGDB_C002833PGDB_AS000209View
2D structure for PGDB_C002848
% Degradation-=60.1%100 nM-CSNK1A1--WO2024059107A1PGDB_A032187PGDB_C002848PGDB_AS000209View
2D structure for PGDB_C002823
% Degradation-=-190.2%100 nM-CSNK1A1--WO2024059107A1PGDB_A032282PGDB_C002823PGDB_AS000209View
2D structure for PGDB_C002807
% Degradation-=12%100 nM-CSNK1A1--WO2024059107A1PGDB_A038385PGDB_C002807PGDB_AS000209View
2D structure for PGDB_C002830
% Degradation-=56.6%100 nM-CSNK1A1--WO2024059107A1PGDB_A038660PGDB_C002830PGDB_AS000209View
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