Activity record

PGDB_A067423

Assay: viabilityTarget: GSPT1QC: ambiguous
Activity overview

GI50 = 2.51 nM

TargetGSPT1
Cell lineSU-DHL-2
Time48 h
Assay / ReadoutGI50 / viability
Assay IDPGDB_AS000205
PatentWO2023237116A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002220
Compound IDPGDB_C002220
CompoundExample 94;Example 94
Source record IDPGDB_C002220
InChIKeyBJZZEXKDIBXDST-YYSPQECZSA-N

Assay context

Assay IDPGDB_AS000205
Assay familyviability
Assay systemcell_based
ReadoutGI50
Treatment time48 h
Detection target% Cell viability
TargetGSPT1
E3Not specified
Cell lineSU-DHL-2

Source evidence

Patent IDWO2023237116A1
Compound location

Example 94;Example 94

Example 94;Example 94 enlarged structureExample 94;Example 94 location on patent page 293
Activity table
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