Assay
PGDB_AS000205
System: cell_basedCell line: SU-DHL-2
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 11.38 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A013438 | PGDB_C002218 | PGDB_AS000205 | View | |
| GI50 | - | = | 4.07 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A036141 | PGDB_C002229 | PGDB_AS000205 | View | |
| GI50 | - | = | 1.3 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A038318 | PGDB_C002285 | PGDB_AS000205 | View | |
| GI50 | - | = | 0.4 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A048801 | PGDB_C002217 | PGDB_AS000205 | View | |
| GI50 | - | = | 1.73 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A057236 | PGDB_C002254 | PGDB_AS000205 | View | |
| GI50 | - | = | 2.24 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A064024 | PGDB_C002231 | PGDB_AS000205 | View | |
| GI50 | - | = | 2.51 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A067423 | PGDB_C002220 | PGDB_AS000205 | View | |
| GI50 | - | = | 0.5 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A077636 | PGDB_C002262 | PGDB_AS000205 | View |