Activity record

PGDB_A067820

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

IC50 = 82 nM

TargetGSPT1
Cell lineMOLM-13
TimeThree days later
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS001125
PatentWO2022073469A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C004693
Compound IDPGDB_C004693
CompoundGS-021;GS-021
Source record IDPGDB_C004693
InChIKeyBLYFAPCZWDYTND-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001125
Assay familyviability
Assay systemcell_based
ReadoutIC50
Treatment timeThree days later
Detection target% Cell viability
TargetGSPT1
E3Not specified
Cell lineMOLM-13

Source evidence

Patent IDWO2022073469A1
Compound location

GS-021;GS-021

GS-021;GS-021 enlarged structureGS-021;GS-021 location on patent page 81
Activity table
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