Assay context summary

Assay context

26 activity records
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C004695
IC50-=3.7nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008880PGDB_C004695PGDB_AS001125View
2D structure for PGDB_C004687
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A009674PGDB_C004687PGDB_AS001125View
2D structure for PGDB_C004685
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A011038PGDB_C004685PGDB_AS001125View
2D structure for PGDB_C004681
IC50-=35nM-GSPT1-MOLM-13WO2022073469A1PGDB_A012386PGDB_C004681PGDB_AS001125View
2D structure for PGDB_C004678
IC50-=29nM-GSPT1-MOLM-13WO2022073469A1PGDB_A012749PGDB_C004678PGDB_AS001125View
2D structure for PGDB_C004688
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A013403PGDB_C004688PGDB_AS001125View
2D structure for PGDB_C004689
IC50-=30nM-GSPT1-MOLM-13WO2022073469A1PGDB_A013891PGDB_C004689PGDB_AS001125View
2D structure for PGDB_C004674
IC50-=583nM-GSPT1-MOLM-13WO2022073469A1PGDB_A020543PGDB_C004674PGDB_AS001125View
2D structure for PGDB_C004676
IC50-=2.1nM-GSPT1-MOLM-13WO2022073469A1PGDB_A021393PGDB_C004676PGDB_AS001125View
2D structure for PGDB_C004673
IC50-=301nM-GSPT1-MOLM-13WO2022073469A1PGDB_A023195PGDB_C004673PGDB_AS001125View
2D structure for PGDB_C004691
IC50-=146nM-GSPT1-MOLM-13WO2022073469A1PGDB_A023340PGDB_C004691PGDB_AS001125View
2D structure for PGDB_C004694
IC50-=875nM-GSPT1-MOLM-13WO2022073469A1PGDB_A025342PGDB_C004694PGDB_AS001125View
2D structure for PGDB_C004698
IC50-=520nM-GSPT1-MOLM-13WO2022073469A1PGDB_A030452PGDB_C004698PGDB_AS001125View
2D structure for PGDB_C004683
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A035108PGDB_C004683PGDB_AS001125View
2D structure for PGDB_C004692
IC50-=87nM-GSPT1-MOLM-13WO2022073469A1PGDB_A037968PGDB_C004692PGDB_AS001125View
2D structure for PGDB_C004696
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A038323PGDB_C004696PGDB_AS001125View
2D structure for PGDB_C004675
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A039047PGDB_C004675PGDB_AS001125View
2D structure for PGDB_C004677
IC50-=11.8nM-GSPT1-MOLM-13WO2022073469A1PGDB_A044484PGDB_C004677PGDB_AS001125View
2D structure for PGDB_C004684
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A045383PGDB_C004684PGDB_AS001125View
2D structure for PGDB_C004697
IC50->10000nM-GSPT1-MOLM-13WO2022073469A1PGDB_A052445PGDB_C004697PGDB_AS001125View