Activity record

PGDB_A069898

Assay: % DegradationTarget: IKZF2QC: standardized
Activity overview

degradation = 82.5 %

TargetIKZF2
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS000892
PatentWO2024059107A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002820
Compound IDPGDB_C002820
Compound72;72;72
Source record IDPGDB_C002820
InChIKeyBUKXXJVKMXZXHH-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000892
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetIKZF2
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

72;72;72

72;72;72 enlarged structure72;72;72 location on patent page 10
Activity table
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