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Compound
PGDB_C002820
8 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)c4ccc5ncsc5c4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 33.2 | % | 100 nM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A021463 | PGDB_C002820 | PGDB_AS000209 | View |
| % Degradation | - | = | 2.7 | % | 100 nM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A038093 | PGDB_C002820 | PGDB_AS000707 | View |
| % Degradation | - | = | 54.5 | % | 1 uM | - | CSNK1A1 | - | - | WO2024059107A1 | PGDB_A040051 | PGDB_C002820 | PGDB_AS000685 | View |
| % Degradation | - | = | -1.7 | % | 100 nM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A042593 | PGDB_C002820 | PGDB_AS002431 | View |
| % Degradation | - | = | -0.9 | % | 1 uM | - | GSPT1 | - | - | WO2024059107A1 | PGDB_A063234 | PGDB_C002820 | PGDB_AS001974 | View |
| % Degradation | - | = | 41.8 | % | 100 nM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A068712 | PGDB_C002820 | PGDB_AS001414 | View |
| % Degradation | - | = | 82.5 | % | 1 uM | - | IKZF2 | - | - | WO2024059107A1 | PGDB_A069898 | PGDB_C002820 | PGDB_AS000892 | View |
| % Degradation | - | = | 6.5 | % | 1 uM | - | IKZF1 | - | - | WO2024059107A1 | PGDB_A072556 | PGDB_C002820 | PGDB_AS000768 | View |