Activity record

PGDB_A071401

Assay: % DegradationTarget: ARQC: ambiguous
Activity overview

degradation = 4 %

TargetAR
Cell lineLNCaP
Concentration2.5 uM
Assay / Readout% Degradation
Assay IDPGDB_AS002020
PatentJP5998117B2
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C026005
Compound IDPGDB_C026005
CompoundASC-Q101
Source record IDPGDB_C026005
InChIKeyBFPWJLYZTCGUIE-QHKWOANTSA-N

Assay context

Assay IDPGDB_AS002020
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration2.5 uM
Detection targetprotein_degradation
TargetAR
E3Not specified
Cell lineLNCaP
OrganismHomo sapiens

Source evidence

Patent IDJP5998117B2
Compound location

ASC-Q101

ASC-Q101 enlarged structureASC-Q101 location on patent page 60
Activity table
Page 70 · table single