Activity record

PGDB_A073790

Assay: % DegradationTarget: CSNK1A1QC: ambiguous
Activity overview

degradation = 25-50 %

TargetCSNK1A1
Concentration0.1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001805
PatentUS20200369679A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C004435
Compound IDPGDB_C004435
CompoundI-5;I-5
Source record IDPGDB_C004435
InChIKeySKAIDPMCBUKTDS-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001805
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration0.1 uM
Detection targetprotein_degradation
TargetCSNK1A1
E3Not specified

Source evidence

Patent IDUS20200369679A1
Compound location

I-5;I-5

I-5;I-5 enlarged structureI-5;I-5 location on patent page 122
Activity table
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