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Compound
PGDB_C004435
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(CNC(=O)C(=O)c4ccc(C5(C(F)(F)F)CC5)cc4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | >= | 80 | % | 1 uM | 3 d | - | - | MOLM-13 | US20200369679A1 | PGDB_A025773 | PGDB_C004435 | PGDB_AS001386 | View |
| % Degradation | - | >= | 80 | % | 0.1 uM | - | GSPT1 | - | - | US20200369679A1 | PGDB_A026459 | PGDB_C004435 | PGDB_AS001685 | View |
| % Degradation | - | >= | 80 | % | 0.1 uM | - | IKZF1 | - | - | US20200369679A1 | PGDB_A059243 | PGDB_C004435 | PGDB_AS002410 | View |
| % Degradation | - | = | 25-50 | % | 0.1 uM | - | CSNK1A1 | - | - | US20200369679A1 | PGDB_A073790 | PGDB_C004435 | PGDB_AS001805 | View |