Activity record

PGDB_A075086

Assay: ternary_complexTarget: RBM39QC: standardized
Activity overview

EC50 < 1 uM

TargetRBM39
E3 ligaseDCAF15
Time1 h
Assay / ReadoutAlphaLISA / EC50
Assay IDPGDB_AS000136
PatentWO2022173805A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009658
Compound IDPGDB_C009658
Compound166
Source record IDPGDB_C009658
InChIKeyJYOIADVAWPZSIY-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000136
Assay familyternary_complex
Assay systembiochemical
ReadoutEC50
TechnologyAlphaLISA
Treatment time1 h
TargetRBM39
E3DCAF15

Source evidence

Patent IDWO2022173805A1
Compound location

166

166 enlarged structure166 location on patent page 150
Activity table
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