Activity record

PGDB_A076418

Assay: bindingQC: standardized_posthoc
Activity overview

selectivity_index <= 100 fold

ControlCDK2 / CDK12
Assay / ReadoutFold change / binding
Assay IDPGDB_AS002325
PatentWO2025110815A1
QC statusstandardized_posthoc
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010901
Compound IDPGDB_C010901
Compound7
Source record IDPGDB_C010901
InChIKeyGYVPSLVCHNWXPK-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002325
Assay familybinding
Assay systemcell_based
ReadoutFold change
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

7

7 enlarged structure7 location on patent page 66
Activity table
Page 154 · table start