Activity record

PGDB_A078259

Assay: biochemicalTarget: CRBNQC: standardized
Activity overview

EC50 = 3.4 uM

TargetCRBN
E3 ligaseCRBN
Assay / ReadoutHTRF / EC50
Assay IDPGDB_AS002171
PatentWO2026099466A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C031219
Compound IDPGDB_C031219
Compound21;21
Source record IDPGDB_C031219
InChIKeyFHXTVTNYXCTQEF-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002171
Assay familybiochemical
Assay systembiochemical
ReadoutEC50
TechnologyHTRF
TargetCRBN
E3CRBN

Source evidence

Patent IDWO2026099466A1
Compound location

21;21

21;21 enlarged structure21;21 location on patent page 53
Activity table
Page 186 · table start
Page 187 · table end