Activity record

PGDB_A079426

Assay: % DegradationTarget: VAV1QC: standardized
Activity overview

Dmax = 99.2 %

TargetVAV1
Time24 h
Assay / Readoutluminescence / Dmax
Assay IDPGDB_AS002286
PatentWO2026098637A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C031198
Compound IDPGDB_C031198
Compound4-2
Source record IDPGDB_C031198
InChIKeyRIFDPWJLHNZGEX-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002286
Assay family% Degradation
Assay systemcell_based
ReadoutDmax
Technologyluminescence
Treatment time24 h
Detection targetprotein_degradation
TargetVAV1
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDWO2026098637A1
Compound location

4-2

4-2 enlarged structure4-2 location on patent page 100
Activity table
Page 99 · table single