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Compound
PGDB_C031198
7 activity records2 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc(-n4ccccc4=O)cc3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 21.55 | nM | - | — | VAV1 | - | - | WO2026114367A1 | PGDB_A001381 | PGDB_C031198 | PGDB_AS000533 | View |
| Dmax | - | = | 98.9 | % | - | 24 h | VAV1 | - | Jurkat | WO2026098637A1 | PGDB_A002233 | PGDB_C031198 | PGDB_AS001360 | View |
| DC50 | - | = | 0.4 | nM | - | — | VAV1 | - | - | WO2026098637A1 | PGDB_A004843 | PGDB_C031198 | PGDB_AS001476 | View |
| DC50 | - | = | 2.8 | nM | - | — | VAV1 | - | Jurkat | WO2026098637A1 | PGDB_A078170 | PGDB_C031198 | PGDB_AS000531 | View |
| Dmax | - | = | 96.5 | % | - | 24 h | VAV1 | - | - | WO2026098637A1 | PGDB_A078779 | PGDB_C031198 | PGDB_AS002175 | View |
| DC50 | - | = | 36.6 | nM | - | — | VAV1 | - | - | WO2026098637A1 | PGDB_A078948 | PGDB_C031198 | PGDB_AS001571 | View |
| Dmax | - | = | 99.2 | % | - | 24 h | VAV1 | - | - | WO2026098637A1 | PGDB_A079426 | PGDB_C031198 | PGDB_AS002286 | View |